BDBM285286 2-[[3-(1,5-dimethyl-6-oxopyridin-3-yl)-5- methylsulfonylphenoxy]methyl]benzonitrile::BDBM486130::US10023592, Example 334
SMILES Cc1cc(cn(C)c1=O)-c1cc(OCc2ccccc2C#N)cc(c1)S(C)(=O)=O
InChI Key InChIKey=JFWHIYWRVFGTSR-UHFFFAOYSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 285286
Affinity DataIC50: <500nMAssay Description:Determination of the IC50 for the heterocyclic derivative BRD4 inhibitors disclosed herein was performed as follows. His-tagged BRD4 was cloned, expr...More data for this Ligand-Target Pair
Affinity DataIC50: <500nMpH: 7.3Assay Description:Determination of the IC50 for the heterocyclic derivative BRD4 inhibitors disclosed herein was performed as follows. His-tagged BRD4 was cloned, expr...More data for this Ligand-Target Pair